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Allosteric modulators restore orthosteric agonist binding to mutated CB(1) receptors

OBJECTIVES: To determine if diminished orthosteric agonist binding due to mutations in extracellular loops 1 or 2 of the cannabinoid receptor 1 (CB(1)) can be overcome by an allosteric modulator and restore agonist binding. METHODS: Binding assays were performed using a range of concentrations of or...

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Publicat a:J Pharm Pharmacol
Autors principals: Dopart, Rachel, Kendall, Debra A
Format: Artigo
Idioma:Inglês
Publicat: Oxford University Press 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6906232/
https://ncbi.nlm.nih.gov/pubmed/31722122
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/jphp.13193
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