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Structural basis for α-bungarotoxin insensitivity of neuronal nicotinic acetylcholine receptors

The ten types of nicotinic acetylcholine receptor α-subunits show substantial sequence homology, yet some types confer high affinity for α-bungarotoxin, whereas others confer negligible affinity. Combining sequence alignments with structural data reveals three residues unique to α-toxin-refractory α...

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Pubblicato in:Neuropharmacology
Autori principali: Sine, Steven M., Strikwerda, John R., Mazzaferro, Simone
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6842095/
https://ncbi.nlm.nih.gov/pubmed/31163179
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.neuropharm.2019.05.037
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