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Synthesis and evaluation of tetrahydropyrazolopyridine inhibitors of anion exchange protein SLC26A4 (pendrin)

Pendrin is a transmembrane chloride/anion antiporter that is strongly upregulated in the airways in rhinoviral infection, asthma, cystic fibrosis and chronic rhinosinusitis. Based on its role in the regulation of airway surface liquid depth, pendrin inhibitors have potential indications for treatmen...

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Détails bibliographiques
Publié dans:Bioorg Med Chem Lett
Auteurs principaux: Zhu, Jie S., Lu, Julia Y., Tan, Joseph-Anthony, Rivera, Amber A., Phuan, Puay-Wah, Shatskikh, Marina E., Son, Jung-Ho, Haggie, Peter M., Verkman, Alan S., Kurth, Mark J.
Format: Artigo
Langue:Inglês
Publié: 2019
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC6690761/
https://ncbi.nlm.nih.gov/pubmed/31281021
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2019.07.003
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