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How to rescue misfolded SERT, DAT and NET: targeting conformational intermediates with atypical inhibitors and partial releasers

Point mutations in the coding sequence for solute carrier 6 (SLC6) family members result in clinically relevant disorders, which are often accounted for by a loss-of-function phenotype. In many instances, the mutated transporter is not delivered to the cell surface because it is retained in the endo...

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Pubblicato in:Biochem Soc Trans
Autori principali: Bhat, Shreyas, Newman, Amy Hauck, Freissmuth, Michael
Natura: Artigo
Lingua:Inglês
Pubblicazione: Portland Press Ltd. 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6599159/
https://ncbi.nlm.nih.gov/pubmed/31064865
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1042/BST20180512
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