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Tropane-Based Ibogaine Analog Rescues Folding-Deficient Serotonin and Dopamine Transporters
[Image: see text] Missense mutations that give rise to protein misfolding are rare, but collectively, defective protein folding diseases are consequential. Folding deficiencies are amenable to pharmacological correction (pharmacochaperoning), but the underlying mechanisms remain enigmatic. Ibogaine...
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| Pubblicato in: | ACS Pharmacol Transl Sci |
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| Autori principali: | , , , , , , , , , , |
| Natura: | Artigo |
| Lingua: | Inglês |
| Pubblicazione: |
American
Chemical Society
2020
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| Accesso online: | https://ncbi.nlm.nih.gov/pmc/articles/PMC8033614/ https://ncbi.nlm.nih.gov/pubmed/33860180 https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsptsci.0c00102 |
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