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Stereoselective Oxidation Kinetics of Deoxycholate in Recombinant and Microsomal CYP3A Enzymes: Deoxycholate 19-Hydroxylation Is an In Vitro Marker of CYP3A7 Activity

The primary bile acids (BAs) synthesized from cholesterol in the liver are converted to secondary BAs by gut microbiota. It was recently disclosed that the major secondary BA, deoxycholate (DCA) species, is stereoselectively oxidized to tertiary BAs exclusively by CYP3A enzymes. This work subsequent...

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Bibliografiske detaljer
Udgivet i:Drug Metab Dispos
Main Authors: Chen, Yu-Jie, Zhang, Jian, Zhu, Ping-Ping, Tan, Xian-Wen, Lin, Qiu-Hong, Wang, Wen-Xia, Yin, Shan-Shan, Gao, Ling-Zhi, Su, Ming-Ming, Liu, Chang-Xiao, Xu, Liang, Jia, Wei, Sevrioukova, Irina F., Lan, Ke
Format: Artigo
Sprog:Inglês
Udgivet: The American Society for Pharmacology and Experimental Therapeutics 2019
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6505377/
https://ncbi.nlm.nih.gov/pubmed/30918015
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.119.086637
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