GABA(A) Receptor Subtype‐Selective Efficacy: TPA023, an α2/α3 Selective Non‐sedating Anxiolytic and α5IA, an α5 Selective Cognition Enhancer

Lignende værker

• Novel Discriminative Stimulus Effects of TPA023B, Subtype-Selective γ-aminobutyric-acid(A)/Benzodiazepine Modulator: Comparisons with Zolpidem, Lorazepam, and TPA023
  af: Kohut, Stephen J., et al.
  Udgivet: (2008)
• 2′-Methoxy-6-methylflavone: a novel anxiolytic and sedative with subtype selective activating and modulating actions at GABA(A) receptors
  af: Karim, Nasiara, et al.
  Udgivet: (2012)
• Reducing Abuse Liability of GABA(A)/Benzodiazepine Ligands via Selective Partial Agonist Efficacy at α(1) and α(2/3) Subtypes
  af: Ator, Nancy A., et al.
  Udgivet: (2010)
• Specific targeting of the GABA-A receptor α5 subtype by a selective inverse agonist restores cognitive deficits in Down syndrome mice
  af: Braudeau, J, et al.
  Udgivet: (2011)
• Analgesic potential of PF-06372865, an α2/α3/α5 subtype-selective GABA(A) partial agonist, in humans
  af: van Amerongen, Guido, et al.
  Udgivet: (2019)