Nalaganje...

Novel Discriminative Stimulus Effects of TPA023B, Subtype-Selective γ-aminobutyric-acid(A)/Benzodiazepine Modulator: Comparisons with Zolpidem, Lorazepam, and TPA023

Anxiolytics with fewer unwanted effects may be created by varying GABAergic efficacy at the BZ binding site across GABA(A) receptor subtypes. TPA023 and TPA023B have in vitro antagonist efficacy at α(1) subtypes and partial-agonist efficacy at α(2/3) subtypes. TPA023B has partial-agonist efficacy at...

Popoln opis

Shranjeno v:
Bibliografske podrobnosti
Main Authors: Kohut, Stephen J., Ator, Nancy A.
Format: Artigo
Jezik:Inglês
Izdano: 2008
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC3010402/
https://ncbi.nlm.nih.gov/pubmed/18395780
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.pbb.2008.02.019
Oznake: Označite
Brez oznak, prvi označite!