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Synthesis and Biological Evaluation of Solithromycin Analogs Against Multidrug Resistant Pathogens

Novel antibacterial drugs that treat multidrug resistant pathogens are in high demand. We have synthesized analogs of solithromycin using Cu(I)-mediated click chemistry. Evaluation of the analogs using Minimum Inhibitory Concentration (MIC) assays against resistant Staphylococcus aureus, Escherichia...

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Detalles Bibliográficos
Publicado en:Bioorg Med Chem Lett
Main Authors: Daher, Samer S., Jin, Xiao, Patel, Jimmy, Freundlich, Joel S., Buttaro, Bettina, Andrade, Rodrigo B.
Formato: Artigo
Idioma:Inglês
Publicado: 2019
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC6487207/
https://ncbi.nlm.nih.gov/pubmed/30962084
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2019.03.038
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