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Structure-Based Virtual Screening and In Vitro Evaluation of New Trypanosoma cruzi Cruzain Inhibitors

Chagas disease (CD), or American trypanosomiasis, causes more than 10,000 deaths per year in the Americas. Current medical therapy for CD has low efficacy in the chronic phase of the disease and serious adverse effects; therefore, it is necessary to search for new pharmacological treatments. In this...

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Dettagli Bibliografici
Pubblicato in:Int J Mol Sci
Autori principali: Herrera-Mayorga, Verónica, Lara-Ramírez, Edgar E., Chacón-Vargas, Karla F., Aguirre-Alvarado, Charmina, Rodríguez-Páez, Lorena, Alcántara-Farfán, Verónica, Cordero-Martínez, Joaquín, Nogueda-Torres, Benjamín, Reyes-Espinosa, Francisco, Bocanegra-García, Virgilio, Rivera, Gildardo
Natura: Artigo
Lingua:Inglês
Pubblicazione: MDPI 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6479639/
https://ncbi.nlm.nih.gov/pubmed/30970549
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/ijms20071742
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