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Intestinal epithelial potassium channels and CFTR chloride channels activated in ErbB tyrosine kinase inhibitor diarrhea

Diarrhea is a major side effect of ErbB receptor tyrosine kinase inhibitors (TKIs) in cancer chemotherapy. Here, we show that the primary mechanism of ErbB TKI diarrhea is activation of basolateral membrane potassium (K(+)) channels and apical membrane chloride (Cl(–)) channels in intestinal epithel...

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Pubblicato in:JCI Insight
Autori principali: Duan, Tianying, Cil, Onur, Thiagarajah, Jay R., Verkman, Alan S.
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Clinical Investigation 2019
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6478423/
https://ncbi.nlm.nih.gov/pubmed/30668547
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1172/jci.insight.126444
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