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THER-29. NOVEL DUAL EGFR/PI3-KINASE INHIBITORS SHOW ENHANCED POTENCY, STRONGER PATHWAY SUPPRESSION AND TARGETING OF METABOLIC PROPERTIES IN PEDIATRIC AND ADULT HIGH GRADE GLIOMA MODELS THAN SINGLE KINASE INHIBITORS

High grade gliomas (HGG), including glioblastoma (GBM) and diffuse intrinsic pontine glioma (DIPG), carry poor prognosis with median survival rates under 15 months post diagnosis. Due to dysregulation of the RTK/PI3K pathways within these tumors, targeted kinase inhibition has been considered a prom...

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Publicado en:Neuro Oncol
Autores principales: Sun, Yusha, Bailey, Cavan, Whitehead, Christopher, Sebolt-Leopold, Judith, Chandra, Joya
Formato: Artigo
Lenguaje:Inglês
Publicado: Oxford University Press 2019
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6477404/
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/neuonc/noz036.234
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