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Efficiency measures the conversion of agonist binding energy into receptor conformational change

Receptors alternate between resting↔active conformations that bind agonists with low↔high affinity. Here, we define a new agonist attribute, energy efficiency (η), as the fraction of ligand-binding energy converted into the mechanical work of the activation conformational change. η depends only on t...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Julkaisussa:J Gen Physiol
Päätekijät: Nayak, Tapan K., Vij, Ridhima, Bruhova, Iva, Shandilya, Jayasha, Auerbach, Anthony
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: Rockefeller University Press 2019
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC6445574/
https://ncbi.nlm.nih.gov/pubmed/30635369
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1085/jgp.201812215
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