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Synthesis and Biochemical Evaluation of Biotinylated Conjugates of Largazole Analogues: Selective Class I Histone Deacetylase Inhibitors

The synthesis of biotinylated conjugates of synthetic analogues of the potent and selective histone deacetylase (HDAC) inhibitor largazole is reported. The thiazole moiety of the parent compound’s cap group was derivatized to allow the chemical conjugation to biotin. The derivatized largazole analog...

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Dettagli Bibliografici
Pubblicato in:Isr J Chem
Autori principali: Zhao, Le, Dunne, Christine E., Clausen, Dane J., Roberts, Justin M., Paulk, Joshiawa, Liu, Haining, Wiest, Olaf G., Bradner, James E., Williams, Robert M.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6370329/
https://ncbi.nlm.nih.gov/pubmed/30760938
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/ijch.201600130
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