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Predicting the Conformational Variability of Abl Tyrosine Kinase using Molecular Dynamics Simulations and Markov State Models

Understanding protein conformational variability remains a challenge in drug discovery. The issue arises in protein kinases, whose multiple conformational states can affect the binding of small-molecule inhibitors. To overcome this challenge, we propose a comprehensive computational framework based...

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Bibliografske podrobnosti
izdano v:J Chem Theory Comput
Main Authors: Meng, Yilin, Gao, Cen, Clawson, David, Atwell, Shane, Russell, Marijane, Vieth, Michal, Roux, Benoît
Format: Artigo
Jezik:Inglês
Izdano: 2018
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC6317529/
https://ncbi.nlm.nih.gov/pubmed/29474075
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jctc.7b01170
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