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The Activation of c-Src Tyrosine Kinase: Conformational Transition Pathway and Free Energy Landscape

Tyrosine kinases are important cellular signaling allosteric enzymes that regulate cell growth, proliferation, metabolism, differentiation and migration. Their activity must be tightly regulated, and disruption of this regulation can lead to a variety of diseases, particularly cancer. The non-recept...

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Pubblicato in:J Phys Chem B
Autori principali: Fajer, Mikolai, Meng, Yilin, Roux, Benoît
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2016
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5398919/
https://ncbi.nlm.nih.gov/pubmed/27715044
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jpcb.6b08409
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