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The Activation of c-Src Tyrosine Kinase: Conformational Transition Pathway and Free Energy Landscape

Tyrosine kinases are important cellular signaling allosteric enzymes that regulate cell growth, proliferation, metabolism, differentiation and migration. Their activity must be tightly regulated, and disruption of this regulation can lead to a variety of diseases, particularly cancer. The non-recept...

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Detalhes bibliográficos
Publicado no:J Phys Chem B
Main Authors: Fajer, Mikolai, Meng, Yilin, Roux, Benoît
Formato: Artigo
Idioma:Inglês
Publicado em: 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5398919/
https://ncbi.nlm.nih.gov/pubmed/27715044
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jpcb.6b08409
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