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The Activation of c-Src Tyrosine Kinase: Conformational Transition Pathway and Free Energy Landscape

Tyrosine kinases are important cellular signaling allosteric enzymes that regulate cell growth, proliferation, metabolism, differentiation and migration. Their activity must be tightly regulated, and disruption of this regulation can lead to a variety of diseases, particularly cancer. The non-recept...

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Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Cyhoeddwyd yn:J Phys Chem B
Prif Awduron: Fajer, Mikolai, Meng, Yilin, Roux, Benoît
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: 2016
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC5398919/
https://ncbi.nlm.nih.gov/pubmed/27715044
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jpcb.6b08409
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