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Stapling of two PEGylated side chains increases the conformational stability of the WW domain via an entropic effect

Hydrocarbon stapling and PEGylation are distinct strategies for enhancing the conformational stability and/or pharmacokinetic properties of peptide and protein drugs. Here we combine these approaches by incorporating asparagine-linked O-allyl PEG oligomers at two positions within the β-sheet protein...

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Detalhes bibliográficos
Publicado no:Org Biomol Chem
Main Authors: Xiao, Qiang, Bécar, Natalie A., Brown, Nathaniel P., Smith, Mason S., Stern, Kimberlee L., Draper, Stven R. E., Thompson, Katherine P., Price, Joshua L.
Formato: Artigo
Idioma:Inglês
Publicado em: 2018
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6290918/
https://ncbi.nlm.nih.gov/pubmed/30444518
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c8ob02535e
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