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Evidence of disulfide bond scrambling during production of an antibody-drug conjugate

Antibody-drug conjugates (ADCs) that are formed using thiol-maleimide chemistry are commonly produced by reactions that occur at or above neutral pHs. Alkaline environments can promote disulfide bond scrambling, and may result in the reconfiguration of interchain disulfide bonds in IgG antibodies, p...

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Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Cyhoeddwyd yn:MAbs
Prif Awduron: Liu-Shin, Lily Pei-Yao, Fung, Adam, Malhotra, Arun, Ratnaswamy, Gayathri
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: Taylor & Francis 2018
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC6284598/
https://ncbi.nlm.nih.gov/pubmed/30339473
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/19420862.2018.1521128
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