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Evidence of disulfide bond scrambling during production of an antibody-drug conjugate

Antibody-drug conjugates (ADCs) that are formed using thiol-maleimide chemistry are commonly produced by reactions that occur at or above neutral pHs. Alkaline environments can promote disulfide bond scrambling, and may result in the reconfiguration of interchain disulfide bonds in IgG antibodies, p...

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Vydáno v:MAbs
Hlavní autoři: Liu-Shin, Lily Pei-Yao, Fung, Adam, Malhotra, Arun, Ratnaswamy, Gayathri
Médium: Artigo
Jazyk:Inglês
Vydáno: Taylor & Francis 2018
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6284598/
https://ncbi.nlm.nih.gov/pubmed/30339473
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/19420862.2018.1521128
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