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Gabapentin Is a Potent Activator of KCNQ3 and KCNQ5 Potassium Channels

Synthetic gabapentinoids, exemplified by gapapentin and pregabalin, are in extensive clinical use for indications including epilepsy, neuropathic pain, anxiety, and alcohol withdrawal. Their mechanisms of action are incompletely understood, but are thought to involve inhibition of α(2)δ subunit–cont...

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Détails bibliographiques
Publié dans:Mol Pharmacol
Auteurs principaux: Manville, Rían W., Abbott, Geoffrey W.
Format: Artigo
Langue:Inglês
Publié: The American Society for Pharmacology and Experimental Therapeutics 2018
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC6108572/
https://ncbi.nlm.nih.gov/pubmed/30021858
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.118.112953
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