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Gabapentin Is a Potent Activator of KCNQ3 and KCNQ5 Potassium Channels

Synthetic gabapentinoids, exemplified by gapapentin and pregabalin, are in extensive clinical use for indications including epilepsy, neuropathic pain, anxiety, and alcohol withdrawal. Their mechanisms of action are incompletely understood, but are thought to involve inhibition of α(2)δ subunit–cont...

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Bibliografske podrobnosti
izdano v:Mol Pharmacol
Main Authors: Manville, Rían W., Abbott, Geoffrey W.
Format: Artigo
Jezik:Inglês
Izdano: The American Society for Pharmacology and Experimental Therapeutics 2018
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC6108572/
https://ncbi.nlm.nih.gov/pubmed/30021858
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.118.112953
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