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Rigid Peptide Macrocycles via On-Resin Glaser Stapling

Peptide macrocycles are widely utilized in the development of high affinity ligands including stapled α-helices. The linear rigidity of a 1,3-diynyl linkage provides an optimal distance (7 Å) between β- carbons of the i, i+4 amino acid side chains, suggesting its utility in stabilizing α-helical str...

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Bibliografiske detaljer
Udgivet i:Chembiochem
Main Authors: Cistrone, Philip A., Silvestri, Anthony P., Hintzen, Jordi C. J., Dawson, Philip E.
Format: Artigo
Sprog:Inglês
Udgivet: 2018
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6097620/
https://ncbi.nlm.nih.gov/pubmed/29516601
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cbic.201800121
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