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Structural bases of TRP channel TRPV6 allosteric modulation by 2-APB

Transient receptor potential (TRP) channels are involved in various physiological processes, including sensory transduction. The TRP channel TRPV6 mediates calcium uptake in epithelia and its expression is dramatically increased in numerous types of cancer. TRPV6 inhibitors suppress tumor growth, bu...

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Publicat a:Nat Commun
Autors principals: Singh, Appu K., Saotome, Kei, McGoldrick, Luke L., Sobolevsky, Alexander I.
Format: Artigo
Idioma:Inglês
Publicat: Nature Publishing Group UK 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6018633/
https://ncbi.nlm.nih.gov/pubmed/29941865
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41467-018-04828-y
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