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Discovery of 2-arylquinazoline derivatives as a new class of ASK1 inhibitors

The development of a new series of apoptosis signal-regulating kinase 1 (ASK1) inhibitors is described. Starting from purine, pyrimidine and quinazoline scaffolds identified by high throughput screening, we used tools of structure-based drug design to develop a series of potent kinase inhibitors, in...

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Detalles Bibliográficos
Publicado en:Bioorg Med Chem Lett
Autores principales: Monastyrskyi, Andrii, Bayle, Simon, Quereda, Victor, Grant, Wayne, Cameron, Michael, Duckett, Derek, Roush, William
Formato: Artigo
Lenguaje:Inglês
Publicado: 2017
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC5999544/
https://ncbi.nlm.nih.gov/pubmed/29277458
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2017.12.026
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