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Optimized allosteric inhibition of engineered protein tyrosine phosphatases with an expanded palette of biarsenical small molecules

Protein tyrosine phosphatases (PTPs), which catalyze the dephosphorylation of phosphotyrosine in protein substrates, are important cell-signaling regulators, as well as potential drug targets for a range of human diseases. Chemical tools for selectively targeting the activities of individual PTPs wo...

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Bibliographic Details
Published in:Bioorg Med Chem
Main Authors: Korntner, Samuel, Pomorski, Adam, Krężel, Artur, Bishop, Anthony C.
Format: Artigo
Language:Inglês
Published: 2018
Subjects:
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC5935566/
https://ncbi.nlm.nih.gov/pubmed/29673715
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2018.04.026
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