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Skp2-dependent reactivation of AKT drives resistance to PI3K inhibitors

The PI3K–AKT kinase signaling pathway is frequently deregulated in human cancers, particularly breast cancer where amplification and somatic mutations of the PIK3CA gene occur with high frequency in patients. Numerous small molecule inhibitors targeting both PI3K and AKT are under clinical evaluatio...

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Detalhes bibliográficos
Publicado no:Sci Signal
Main Authors: Clement, Emilie, Inuzuka, Hiroyuki, Nihira, Naoe T., Wei, Wenyi, Toker, Alex
Formato: Artigo
Idioma:Inglês
Publicado em: 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5902813/
https://ncbi.nlm.nih.gov/pubmed/29535262
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1126/scisignal.aao3810
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