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Skp2-dependent reactivation of AKT drives resistance to PI3K inhibitors

The PI3K–AKT kinase signaling pathway is frequently deregulated in human cancers, particularly breast cancer where amplification and somatic mutations of the PIK3CA gene occur with high frequency in patients. Numerous small molecule inhibitors targeting both PI3K and AKT are under clinical evaluatio...

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Détails bibliographiques
Publié dans:Sci Signal
Auteurs principaux: Clement, Emilie, Inuzuka, Hiroyuki, Nihira, Naoe T., Wei, Wenyi, Toker, Alex
Format: Artigo
Langue:Inglês
Publié: 2018
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5902813/
https://ncbi.nlm.nih.gov/pubmed/29535262
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1126/scisignal.aao3810
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