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Skp2-dependent reactivation of AKT drives resistance to PI3K inhibitors

The PI3K–AKT kinase signaling pathway is frequently deregulated in human cancers, particularly breast cancer where amplification and somatic mutations of the PIK3CA gene occur with high frequency in patients. Numerous small molecule inhibitors targeting both PI3K and AKT are under clinical evaluatio...

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Bibliografski detalji
Izdano u:Sci Signal
Glavni autori: Clement, Emilie, Inuzuka, Hiroyuki, Nihira, Naoe T., Wei, Wenyi, Toker, Alex
Format: Artigo
Jezik:Inglês
Izdano: 2018
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5902813/
https://ncbi.nlm.nih.gov/pubmed/29535262
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1126/scisignal.aao3810
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