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Species differences in drug glucuronidation: Humanized UDP-glucuronosyltransferase 1 mice and their application for predicting drug glucuronidation and drug-induced toxicity in humans

More than 20% of clinically used drugs are glucuronidated by a microsomal enzyme UDP-glucuronosyltransferase (UGT). Inhibition or induction of UGT can result in an increase or decrease in blood drug concentration. To avoid drug-drug interactions and adverse drug reactions in individuals, therefore,...

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Detalhes bibliográficos
Publicado no:Drug Metab Pharmacokinet
Main Authors: Fujiwara, Ryoichi, Yoda, Emiko, Tukey, Robert H.
Formato: Artigo
Idioma:Inglês
Publicado em: 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5809266/
https://ncbi.nlm.nih.gov/pubmed/29079228
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.dmpk.2017.10.002
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