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Glucuronidation of Drugs and Drug-Induced Toxicity in Humanized UDP-Glucuronosyltransferase 1 Mice

UDP-glucuronosyltransferases (UGTs) are phase II drug-metabolizing enzymes that catalyze glucuronidation of various drugs. Although experimental rodents are used in preclinical studies to predict glucuronidation and toxicity of drugs in humans, species differences in glucuronidation and drug-induced...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Egile Nagusiak: Kutsuno, Yuki, Itoh, Tomoo, Tukey, Robert H., Fujiwara, Ryoichi
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: The American Society for Pharmacology and Experimental Therapeutics 2014
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC4053997/
https://ncbi.nlm.nih.gov/pubmed/24764149
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.114.057083
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