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Pharmacologic Evidence for a Putative Conserved Allosteric Site on Opioid Receptors

Allosteric modulators of G protein–coupled receptors, including opioid receptors, have been proposed as possible therapeutic agents with enhanced selectivity. BMS-986122 is a positive allosteric modulator (PAM) of the μ-opioid receptor (µ-OR). BMS-986187 is a structurally distinct PAM for the δ-opio...

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Bibliografski detalji
Izdano u:Mol Pharmacol
Glavni autori: Livingston, Kathryn E., Stanczyk, M. Alexander, Burford, Neil T., Alt, Andrew, Canals, Meritxell, Traynor, John R.
Format: Artigo
Jezik:Inglês
Izdano: The American Society for Pharmacology and Experimental Therapeutics 2018
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5767684/
https://ncbi.nlm.nih.gov/pubmed/29233847
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/mol.117.109561
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