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Atomic view of the energy landscape in the allosteric regulation of Abl kinase

The activity of protein kinases is often regulated in an intramolecular fashion by signaling domains, which feature several phosphorylation or protein-docking sites. How kinases integrate such distinct binding and signaling events to regulate their activities is unclear, especially in quantitative t...

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Библиографические подробности
Опубликовано в: :Nat Struct Mol Biol
Главные авторы: Saleh, Tamjeed, Rossi, Paolo, Kalodimos, Charalampos G.
Формат: Artigo
Язык:Inglês
Опубликовано: 2017
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC5745040/
https://ncbi.nlm.nih.gov/pubmed/28945248
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nsmb.3470
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