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Atomic view of the energy landscape in the allosteric regulation of Abl kinase

The activity of protein kinases is often regulated in an intramolecular fashion by signaling domains, which feature several phosphorylation or protein-docking sites. How kinases integrate such distinct binding and signaling events to regulate their activities is unclear, especially in quantitative t...

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Detalles Bibliográficos
Publicado en:Nat Struct Mol Biol
Main Authors: Saleh, Tamjeed, Rossi, Paolo, Kalodimos, Charalampos G.
Formato: Artigo
Idioma:Inglês
Publicado: 2017
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5745040/
https://ncbi.nlm.nih.gov/pubmed/28945248
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nsmb.3470
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