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Design and Synthesis of N1-Modified Imidazoquinoline Agonists for Selective Activation of Toll-like Receptors 7 and 8

[Image: see text] A series of N1-modified imidazoquinolines were synthesized and screened for Toll-like receptors (TLR) 7 and 8 activities to identify recognition elements that confer high affinity binding and selectivity. These receptors are key targets in the development of immunomodulatory agents...

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Опубликовано в: :ACS Med Chem Lett
Главные авторы: Larson, Peter, Kucaba, Tamara A., Xiong, Zhengming, Olin, Michael, Griffith, Thomas S., Ferguson, David M.
Формат: Artigo
Язык:Inglês
Опубликовано: American Chemical Society 2017
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC5683703/
https://ncbi.nlm.nih.gov/pubmed/29152046
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.7b00256
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