A Direct In Vivo Comparison of The Melanocortin Monovalent Agonist Ac-His-DPhe-Arg-Trp-NH(2) versus The Bivalent Agonist Ac-His-DPhe-Arg-Trp-PEDG20-His-DPhe-Arg-Trp-NH(2): A Bivalent Advantage

Gelijkaardige items

• Synthesis and Pharmacology of α/β(3)-Peptides Based on the Melanocortin Agonist Ac-His-dPhe-Arg-Trp-NH(2) Sequence
  door: Singh, Anamika, et al.
  Gepubliceerd in: (2015)
• Discovery of melanocortin ligands via a double simultaneous substitution strategy based on the Ac-His-DPhe-Arg-Trp-NH(2) template
  door: Todorovic, Aleksandar, et al.
  Gepubliceerd in: (2018)
• Melanocortin Tetrapeptide Ac-His-DPhe-Arg-Trp-NH(2) Modified at the Para Position of the Benzyl Side Chain (DPhe): Importance for Mouse Melanocortin-3 Receptor Agonist versus Antagonist Activity
  door: Proneth, Bettina, et al.
  Gepubliceerd in: (2008)
• The Ac-Trp-DPhe(p-I)-Arg-Trp-NH(2) 250-Fold Selective Melanocortin-4 Receptor (MC4R) Antagonist over the Melanocortin-3 Receptor (MC3R) Affects Energy Homeostasis in Male and Female Mice Differently
  door: Lensing, Cody J., et al.
  Gepubliceerd in: (2016)
• Comparative intracerebroventricular (ICV) and intrathecal (IT) administration of a nanomolar macrocyclic melanocortin receptor agonist MDE6-5-2c (c[Pro-His-DPhe-Arg-Trp-Dap-Ala-DPro]) decreases food intake in mice.
  door: Adank, Danielle N., et al.
  Gepubliceerd in: (2020)