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Design, Synthesis, and Structure–Activity Relationships of Pyrimido[4,5-b]indole-4-amines as Microtubule Depolymerizing Agents that are Effective against Multidrug Resistant Cells

To identify the structural features of 9H-pyrimido[4,5-b]indoles as microtubule depolymerizers, pyrimido[4,5-b]indoles 2–8 with varied substituents at the 2-, 4- and 5-positions were designed and synthesized. Nucleophilic displacement of 2,5-substituted-4-chloro- pyrimido[4,5-b]indoles with appropri...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem Lett
Main Authors: Devambatla, Ravi Kumar Vyas, Li, Wei, Zaware, Nilesh, Choudhary, Shruti, Hamel, Ernest, Mooberry, Susan L., Gangjee, Aleem
Formato: Artigo
Idioma:Inglês
Publicado em: 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5603926/
https://ncbi.nlm.nih.gov/pubmed/28610978
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2017.05.085
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