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Structure-activity relationship studies of G9a-like protein (GLP) inhibitors

Given the high homology between the protein lysine methyltransferases G9a-like protein (GLP) and G9a, it has been challenging to develop potent and selective inhibitors for either enzyme. Recently, we reported two quinazoline compounds, MS0124 and MS012, as GLP selective inhibitors. To further inves...

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Библиографические подробности
Опубликовано в: :Bioorg Med Chem
Главные авторы: Xiong, Yan, Li, Fengling, Babault, Nicolas, Wu, Hong, Dong, Aiping, Zeng, Hong, Chen, Xin, Arrowsmith, Cheryl H., Brown, Peter J., Liu, Jing, Vedadi, Masoud, Jin, Jian
Формат: Artigo
Язык:Inglês
Опубликовано: 2017
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC5562403/
https://ncbi.nlm.nih.gov/pubmed/28662962
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2017.06.021
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