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Identification of 2,4-diamino-6,7-dimethoxyquinoline derivatives as G9a inhibitors

G9a is a histone lysine methyltransferase (HKMT) involved in epigenetic regulation via the installation of histone methylation marks. 6,7-Dimethoxyquinazoline analogues, such as BIX-01294, are established as potent, substrate competitive inhibitors of G9a. With an objective to identify novel chemoty...

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Vydáno v:Medchemcomm
Hlavní autoři: Srimongkolpithak, Nitipol, Sundriyal, Sandeep, Li, Fengling, Vedadi, Masoud, Fuchter, Matthew J.
Médium: Artigo
Jazyk:Inglês
Vydáno: Royal Society of Chemistry 2014
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC4349132/
https://ncbi.nlm.nih.gov/pubmed/25750706
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/c4md00274a
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