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Design of benzoxathiazin-3-one 1,1-dioxides as a new class of irreversible serine hydrolase inhibitors: discovery of a uniquely selective PNPLA4 inhibitor

The design and examination of 4,1,2-benzoxathiazin-3-one 1,1-dioxides as candidate serine hydrolase inhibitors are disclosed, and represent the synthesis and study of a previously unexplored heterocycle. This new class of activated cyclic carbamates provided selective irreversible inhibition of a sm...

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Bibliografische gegevens
Gepubliceerd in:J Am Chem Soc
Hoofdauteurs: Kornahrens, Anne F., Cognetta, Armand B., Brody, Daniel M., Matthews, Megan L., Cravatt, Benjamin F., Boger, Dale L.
Formaat: Artigo
Taal:Inglês
Gepubliceerd in: 2017
Onderwerpen:
Online toegang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5501285/
https://ncbi.nlm.nih.gov/pubmed/28498651
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jacs.7b02985
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