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Proteome-wide reactivity profiling identifies diverse carbamate chemotypes tuned for serine hydrolase inhibition

Serine hydrolases are one of the largest and most diverse enzyme classes in Nature. Inhibitors of serine hydrolases are used to treat many diseases, including obesity, diabetes, cognitive dementia, and bacterial and viral infections. Nonetheless, the majority of the 200+ serine hydrolases in mammals...

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Autori principali: Chang, Jae Won, Cognetta, Armand B., Niphakis, Micah J., Cravatt, Benjamin F.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2013
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC3806897/
https://ncbi.nlm.nih.gov/pubmed/23701408
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/cb400261h
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