Carregant...

N-Acyl pyrazoles: effective and tunable inhibitors of serine hydrolases

A series of N-acyl pyrazoles was examined as candidate serine hydrolase inhibitors in which the active site acylating reactivity and the leaving group ability of the pyrazole could be tuned not only through the nature of the acyl group (reactivity: amide > carbamate > urea), but also through p...

Descripció completa

Guardat en:
Dades bibliogràfiques
Publicat a:Bioorg Med Chem
Autors principals: Otrubova, Katerina, Chatterjee, Shreyosree, Ghimire, Srijana, Cravatt, Benjamin F., Boger, Dale L.
Format: Artigo
Idioma:Inglês
Publicat: 2019
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6474344/
https://ncbi.nlm.nih.gov/pubmed/30879861
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2019.03.020
Etiquetes: Afegir etiqueta
Sense etiquetes, Sigues el primer a etiquetar aquest registre!