Nalaganje...

N-Acyl pyrazoles: effective and tunable inhibitors of serine hydrolases

A series of N-acyl pyrazoles was examined as candidate serine hydrolase inhibitors in which the active site acylating reactivity and the leaving group ability of the pyrazole could be tuned not only through the nature of the acyl group (reactivity: amide > carbamate > urea), but also through p...

Popoln opis

Shranjeno v:
Bibliografske podrobnosti
izdano v:Bioorg Med Chem
Main Authors: Otrubova, Katerina, Chatterjee, Shreyosree, Ghimire, Srijana, Cravatt, Benjamin F., Boger, Dale L.
Format: Artigo
Jezik:Inglês
Izdano: 2019
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC6474344/
https://ncbi.nlm.nih.gov/pubmed/30879861
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2019.03.020
Oznake: Označite
Brez oznak, prvi označite!