A carregar...

N-Acyl pyrazoles: effective and tunable inhibitors of serine hydrolases

A series of N-acyl pyrazoles was examined as candidate serine hydrolase inhibitors in which the active site acylating reactivity and the leaving group ability of the pyrazole could be tuned not only through the nature of the acyl group (reactivity: amide > carbamate > urea), but also through p...

ver descrição completa

Na minha lista:
Detalhes bibliográficos
Publicado no:Bioorg Med Chem
Main Authors: Otrubova, Katerina, Chatterjee, Shreyosree, Ghimire, Srijana, Cravatt, Benjamin F., Boger, Dale L.
Formato: Artigo
Idioma:Inglês
Publicado em: 2019
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6474344/
https://ncbi.nlm.nih.gov/pubmed/30879861
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2019.03.020
Tags: Adicionar Tag
Sem tags, seja o primeiro a adicionar uma tag!