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N-Acyl pyrazoles: effective and tunable inhibitors of serine hydrolases

A series of N-acyl pyrazoles was examined as candidate serine hydrolase inhibitors in which the active site acylating reactivity and the leaving group ability of the pyrazole could be tuned not only through the nature of the acyl group (reactivity: amide > carbamate > urea), but also through p...

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Библиографические подробности
Опубликовано в: :Bioorg Med Chem
Главные авторы: Otrubova, Katerina, Chatterjee, Shreyosree, Ghimire, Srijana, Cravatt, Benjamin F., Boger, Dale L.
Формат: Artigo
Язык:Inglês
Опубликовано: 2019
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC6474344/
https://ncbi.nlm.nih.gov/pubmed/30879861
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2019.03.020
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