Yüklüyor......

Design of benzoxathiazin-3-one 1,1-dioxides as a new class of irreversible serine hydrolase inhibitors: discovery of a uniquely selective PNPLA4 inhibitor

The design and examination of 4,1,2-benzoxathiazin-3-one 1,1-dioxides as candidate serine hydrolase inhibitors are disclosed, and represent the synthesis and study of a previously unexplored heterocycle. This new class of activated cyclic carbamates provided selective irreversible inhibition of a sm...

Ful tanımlama

Kaydedildi:
Detaylı Bibliyografya
Yayımlandı:J Am Chem Soc
Asıl Yazarlar: Kornahrens, Anne F., Cognetta, Armand B., Brody, Daniel M., Matthews, Megan L., Cravatt, Benjamin F., Boger, Dale L.
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: 2017
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC5501285/
https://ncbi.nlm.nih.gov/pubmed/28498651
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/jacs.7b02985
Etiketler: Etiketle
Etiket eklenmemiş, İlk siz ekleyin!