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Disulfide trapping to localize small-molecule agonists and antagonists for a G protein-coupled receptor

A key question regarding the signaling mechanism for G protein-coupled receptors (GPCRs) is what triggers agonism versus antagonism. Peptide analogs derived from the chemokine, complement fragment 5 anaphylatoxin (C5a), can act as agonists or antagonists to the C5a receptor, a member of the GPCR fam...

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Autors principals: Buck, Elizabeth, Wells, James A.
Format: Artigo
Idioma:Inglês
Publicat: National Academy of Sciences 2005
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC549436/
https://ncbi.nlm.nih.gov/pubmed/15710877
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.0500016102
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