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Benzimidazole inhibitors from the Niclosamide chemotype inhibit Wnt/β-catenin signaling with selectivity over effects on ATP homeostasis

The Wnt signaling pathway plays a key role in organ and tissue homeostasis, and when dysregulated, can become a major underlying mechanism of disease, particularly cancer. We reported previously that the anthelmintic drug Niclosamide inhibits Wnt/β-catenin signaling and suppresses colon cancer cell...

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Foilsithe in:Bioorg Med Chem
Main Authors: Mook, Robert A., Ren, Xiu-Rong, Wang, Jiangbo, Piao, Hailan, Barak, Larry S., Lyerly, H. Kim, Chen, Wei
Formáid: Artigo
Teanga:Inglês
Foilsithe: 2017
Ábhair:
Rochtain Ar Líne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5490664/
https://ncbi.nlm.nih.gov/pubmed/28233680
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2017.01.046
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