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Peripherally Selective Cannabinoid 1 Receptor (CB1R) Agonists for the Treatment of Neuropathic Pain

Alleviation of neuropathic pain by cannabinoids is limited by their central nervous system (CNS) side effects. Indole and indene compounds were engineered for high hCB1R affinity, peripheral selectivity, metabolic stability, and in vivo efficacy. An epithelial cell line assay identified candidates w...

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Bibliografski detalji
Izdano u:J Med Chem
Glavni autori: Seltzman, Herbert H., Shiner, Craig, Hirt, Erin E., Gilliam, Anne F., Thomas, Brian F., Maitra, Rangan, Snyder, Rod, Black, Sherry L., Patel, Purvi R., Mulpuri, Yatendra, Spigelman, Igor
Format: Artigo
Jezik:Inglês
Izdano: 2016
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5474949/
https://ncbi.nlm.nih.gov/pubmed/27482723
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.6b00516
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