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Peripherally Selective Cannabinoid 1 Receptor (CB1R) Agonists for the Treatment of Neuropathic Pain

Alleviation of neuropathic pain by cannabinoids is limited by their central nervous system (CNS) side effects. Indole and indene compounds were engineered for high hCB1R affinity, peripheral selectivity, metabolic stability, and in vivo efficacy. An epithelial cell line assay identified candidates w...

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Detalhes bibliográficos
Publicado no:J Med Chem
Main Authors: Seltzman, Herbert H., Shiner, Craig, Hirt, Erin E., Gilliam, Anne F., Thomas, Brian F., Maitra, Rangan, Snyder, Rod, Black, Sherry L., Patel, Purvi R., Mulpuri, Yatendra, Spigelman, Igor
Formato: Artigo
Idioma:Inglês
Publicado em: 2016
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Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5474949/
https://ncbi.nlm.nih.gov/pubmed/27482723
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jmedchem.6b00516
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