Načítá se...

Lysosome-oriented, dual-stage pH-responsive polymeric micelles for β-Lapachone delivery

β-Lapachone (β-lap), a novel anticancer agent, is bioactivated by NADP(H):quinone oxidoreductase 1 (NQO1), an enzyme over-expressed in numerous tumors, including lung, pancreas, breast, and prostate cancers. Fast renal clearance and methemaglobinemia / hemolytic side-effects from the clinical formul...

Celý popis

Uloženo v:
Podrobná bibliografie
Vydáno v:J Mater Chem B Mater Biol Med
Hlavní autoři: Zhou, Yinjian, Dong, Ying, Huang, Gang, Wang, Yiguang, Huang, Xiaonan, Zhang, Fayun, Boothman, David A., Gao, Jinming, Liang, Wei
Médium: Artigo
Jazyk:Inglês
Vydáno: 2016
Témata:
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5452003/
https://ncbi.nlm.nih.gov/pubmed/28580145
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/C6TB02049F
Tagy: Přidat tag
Žádné tagy, Buďte první, kdo otaguje tento záznam!