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Lysosome-oriented, dual-stage pH-responsive polymeric micelles for β-Lapachone delivery

β-Lapachone (β-lap), a novel anticancer agent, is bioactivated by NADP(H):quinone oxidoreductase 1 (NQO1), an enzyme over-expressed in numerous tumors, including lung, pancreas, breast, and prostate cancers. Fast renal clearance and methemaglobinemia / hemolytic side-effects from the clinical formul...

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Dades bibliogràfiques
Publicat a:J Mater Chem B Mater Biol Med
Autors principals: Zhou, Yinjian, Dong, Ying, Huang, Gang, Wang, Yiguang, Huang, Xiaonan, Zhang, Fayun, Boothman, David A., Gao, Jinming, Liang, Wei
Format: Artigo
Idioma:Inglês
Publicat: 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5452003/
https://ncbi.nlm.nih.gov/pubmed/28580145
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1039/C6TB02049F
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