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Prodrug Strategy to Achieve Lyophilizable, High Drug Loading Micelle Formulations Through Diester Derivatives of β-Lapachone

β-Lap prodrug micelle strategy improve the formulation properties of β-lap therapeutics. The resulting micelles yielded apparent high β-lap solubility (>7 mg/mL), physical stability, and ability to reconstitute after lyophilization. In the presence of esterase, β-lap prodrugs were efficiently con...

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Autori principali: Ma, Xinpeng, Huang, Xiumei, Huang, Gang, Li, Longshan, Wang, Yiguang, Luo, Xiuquan, Boothman, David A., Gao, Jinming
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2014
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC4133338/
https://ncbi.nlm.nih.gov/pubmed/24532286
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/adhm.201300590
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