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Benzimidazole Analogs as Potent Hypoxia Inducible Factor Inhibitors: Synthesis, Biological Evaluation, and Profiling Drug-like Properties

AIM: To develop potent HIF-1α inhibitors for potential treatment of cancer. MATERIALS AND METHODS: Chemical synthesis, HIF-luciferase assay, cytotoxic assay, platelet aggregation assay, western blot analysis, quantitative real-time PCR, aqueous solubility, protein binding, metabolic stability, and m...

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Salvato in:
Dettagli Bibliografici
Pubblicato in:Anticancer Res
Autori principali: Chen, Jianjun, Wang, Jin, Schwab, Luciana P., Park, Kyung-Tae, Seagroves, Tiffany N., Jennings, Lisa K., Miller, Duane D., Li, Wei
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2014
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5346463/
https://ncbi.nlm.nih.gov/pubmed/25075010
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